BDBM50661339 CHEMBL6147364

SMILES CS(=N)(=O)c1cccc(NC(=O)c2cc(C(F)(F)F)cnc2Oc2ccc(F)cc2Cl)c1

InChI Key InChIKey=YTTNKXUAJRPSAF-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50661339   

TargetSodium channel protein type 10 subunit alpha(Human)
Lieber Institute for Brain Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661339BDBM50661339(CHEMBL6147364)
Affinity DataIC50: 12nMAssay Description:Inhibition of human Nav1.8 with resting membrane potential at half inactivated state by PatchXpress high-throughput electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetSodium channel protein type 10 subunit alpha(Human)
Lieber Institute for Brain Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661339BDBM50661339(CHEMBL6147364)
Affinity DataIC50: 43nMAssay Description:Inhibition of human Nav1.8 with resting membrane potential by PatchXpress high-throughput electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetSodium channel protein type 10 subunit alpha(Mouse)
Lieber Institute for Brain Development

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50661339BDBM50661339(CHEMBL6147364)
Affinity DataIC50: 660nMAssay Description:Inhibition of mouse Nav1.8 with resting membrane potential at half inactivated state by PatchXpress high-throughput electrophysiology methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed