BDBM50662330 CHEMBL6162165
SMILES CCn1c(cc(n1)C(=O)Nc2cccc(c2)NS(=O)(=O)C)C
InChI Key InChIKey=RNCRRFDHODBLRY-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50662330
Affinity DataKd: 330nMAssay Description:Binding affinity to human DHX9 assessed as dissociation constant measured for 360 sec by SPR analysisMore data for this Ligand-Target Pair
Affinity DataKd: 400nMAssay Description:Binding affinity to human DHX9 assessed as dissociation constant measured for 360 sec in presence of ATP by SPR analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 2.90E+3nMAssay Description:Inhibition of human DHX9 using double-stranded RNA and ATP as substrate pre-incubated for 15 mins followed by substrate addition and measured after 6...More data for this Ligand-Target Pair
Affinity DataIC50: 2.14E+4nMAssay Description:Inhibition of human DHX9 using split-beacon oligonucleotide and ATP as substrate pre-incubated for 15 mins followed by substrate addition and measure...More data for this Ligand-Target Pair
Affinity DataEC50: >3.00E+4nMAssay Description:Inhibition of DHX9 in human PBMC assessed as target engagement by measuring circBRIP1 incubated for 24 hrs by Taqman qPCR analysisMore data for this Ligand-Target Pair

3D Structure (crystal)