BDBM50663373 CHEMBL562641

SMILES CCc1ccccc1-c1cccc2[nH]c(C(=O)NC[C@@H](N)C(=O)O)cc12

InChI Key InChIKey=OQLODOGGOMSJDF-UHFFFAOYSA-N

Data  8 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 50663373   

TargetGlutamate NMDA receptor; Grin1/Grin2c(Rat)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50663373BDBM50663373(CHEMBL562641)
Affinity DataEC50:  1nMAssay Description:Agonist activity at recombinant rat GluN1/GluN2C NMDA receptor expressed in xenopus laevis oocytes in presence of glutamate by two-electrode voltage-...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetIonotropic glutamate receptor NMDA 1/2C(Human)
H. Lundbeck A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50663373BDBM50663373(CHEMBL562641)
Affinity DataEC50:  3nMAssay Description:Partial agonist activity at recombinant wild-type human GluN1/2C expressed in Xenopus laevis oocytes by TEVC recording methodMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50663373BDBM50663373(CHEMBL562641)
Affinity DataEC50:  14nMAssay Description:Agonist activity at recombinant rat GluN1/GluN2B NMDA receptor expressed in xenopus laevis oocytes in presence of glutamate by two-electrode voltage-...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetIonotropic glutamate receptor NMDA 1/2D(Rat)
H. Lundbeck A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50663373BDBM50663373(CHEMBL562641)
Affinity DataEC50:  25nMAssay Description:Partial agonist activity at recombinant wild-type human GluN1/2D expressed in Xenopus laevis oocytes by TEVC recording methodMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50663373BDBM50663373(CHEMBL562641)
Affinity DataEC50:  25nMAssay Description:Partial agonist activity at recombinant wild-type human GluN1/2B expressed in Xenopus laevis oocytes by TEVC recording methodMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetIonotropic glutamate receptor NMDA 1/2D(Rat)
H. Lundbeck A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50663373BDBM50663373(CHEMBL562641)
Affinity DataEC50:  31nMAssay Description:Agonist activity at recombinant rat GluN1/GluN2D NMDA receptor expressed in xenopus laevis oocytes in presence of glutamate by two-electrode voltage-...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Human)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50663373BDBM50663373(CHEMBL562641)
Affinity DataEC50:  36nMAssay Description:Agonist activity at recombinant rat GluN1/GluN2A NMDA receptor expressed in xenopus laevis oocytes in presence of glutamate by two-electrode voltage-...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/5/2026
Entry Details
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Human)
University of Copenhagen

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50663373BDBM50663373(CHEMBL562641)
Affinity DataEC50:  66nMAssay Description:Partial agonist activity at recombinant wild-type human GluN1/2A expressed in Xenopus laevis oocytes by TEVC recording methodMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed