BDBM50664814 CHEMBL6146530

SMILES CCc1oncc1-c1cc(F)cc(C(=O)NC[C@@H](N)C(=O)O)c1

InChI Key InChIKey=SFERCLORGFKWPI-UHFFFAOYSA-N

Data  1 KI  4 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50664814   

TargetGlutamate receptor ionotropic, NMDA 1(Human)
H. Lundbeck A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664814BDBM50664814(CHEMBL6146530)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]-MDL105519 from GluN1 LBD (unknown origin) incubated for 30 mins by SPAMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2A(Human)
H. Lundbeck A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664814BDBM50664814(CHEMBL6146530)
Affinity DataEC50:  240nMAssay Description:Agonist activity at recombinant human GluN1/2A expressed in Xenopus laevis oocytes by TEVC recording methodMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetGlutamate receptor ionotropic, NMDA 1/2B(Human)
H. Lundbeck A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664814BDBM50664814(CHEMBL6146530)
Affinity DataEC50:  310nMAssay Description:Agonist activity at recombinant human GluN1/2B expressed in Xenopus laevis oocytes by TEVC recording methodMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetIonotropic glutamate receptor NMDA 1/2C(Human)
H. Lundbeck A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664814BDBM50664814(CHEMBL6146530)
Affinity DataEC50:  360nMAssay Description:Agonist activity at recombinant human GluN1/2C expressed in Xenopus laevis oocytes by TEVC recording methodMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed
TargetIonotropic glutamate receptor NMDA 1/2D(Rat)
H. Lundbeck A/S

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50664814BDBM50664814(CHEMBL6146530)
Affinity DataEC50:  530nMAssay Description:Agonist activity at recombinant human GluN1/2D expressed in Xenopus laevis oocytes by TEVC recording methodMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
6/6/2026
Entry Details
PubMed