BDBM514131 US11052091, Example 5-8

SMILES COc1cc(ccc1Nc1nc(N)c2n(-c3ccc4cn[nH]c4c3)c(=O)n(C3CCOC3)c2n1)S(C)(=O)=O

InChI Key InChIKey=AWLMRYOSUVGNRO-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 514131   

TargetProtein-tyrosine kinase 6(Human)
Ono Pharmaceutical

US Patent
LigandPNGBDBM514131(US11052091, Example 5-8)
Affinity DataIC50: 9nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2022
Entry Details
US Patent