BDBM514138 US11052091, Example 5-21

SMILES COc1cc(Nc2nc(N)c3n(-c4ccc5[nH]ccc5c4)c(=O)n(C(C)C)c3n2)ccc1C(=O)N(C)C

InChI Key InChIKey=XTXTYBRORYAUIJ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 514138   

TargetProtein-tyrosine kinase 6(Human)
Ono Pharmaceutical

US Patent
LigandPNGBDBM514138(US11052091, Example 5-21)
Affinity DataIC50: 5nMAssay Description:Measurement of an inhibitory activity on Brk enzyme was performed by using LanthaScreen (registered trademark) system (Invitrogen) in accordance with...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/6/2022
Entry Details
US Patent