BDBM523797 US11136312, Compound AH.2.178

SMILES Fc1ccc2c(Cc3nnc(SCc4ccccc4)n3CCCc3c[nH]cn3)c[nH]c2c1

InChI Key InChIKey=MOEFJXQMDNBDGY-UHFFFAOYSA-N

Data  2 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 523797   

TargetSomatostatin receptor type 4(Homo sapiens (Human))
Board of Trustees of The Southern Illinois University

US Patent
LigandPNGBDBM523797(US11136312, Compound AH.2.178)
Affinity DataKi:  12.3nMAssay Description:Competitive radioligand binding experiments were performed using MEMBRANE TARGET Systems (Perkin-Elmer, Boston, Mass.) for human somatostatin recepto...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Board of Trustees of The Southern Illinois University

US Patent
LigandPNGBDBM523797(US11136312, Compound AH.2.178)
Affinity DataKi: >1.00E+4nMAssay Description:Competitive radioligand binding experiments were performed using MEMBRANE TARGET Systems (Perkin-Elmer, Boston, Mass.) for human somatostatin recepto...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Board of Trustees of The Southern Illinois University

US Patent
LigandPNGBDBM523797(US11136312, Compound AH.2.178)
Affinity DataEC50:  17.5nMAssay Description:Measurement of forskolin stimulated inhibition of cAMP was performed via time-resolved fluorescence resonance energy transfer (TR-FRET) LANCE assay (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent