BDBM537057 US11897851, Compound 154

SMILES CC1(Oc2cccc(C3CCN(CC4NC=C(\C=C\C(O)=O)N4C[C@H]4CCOC4)CC3)c2O1)c1ccc(Cl)cc1F

InChI Key InChIKey=KETJVXFAJCSPME-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 537057   

TargetGlucagon-like peptide 1 receptor(Human)
Gasherbrum Bio

US Patent
LigandPNGBDBM537057(US11897851, Compound 154)
Affinity DataEC50:  0.0120nMAssay Description:To optimize functional activity directed toward Gas coupling, a HEK293/CRE-Luc cell line developed by HDB stably expressing the GLP-1 Receptor was us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2024
Entry Details
US Patent