BDBM556452 US11897851, Compound 208a

SMILES CCn1cncc1Cn1c(CN2CCC(CC2)c2cccc3O[C@@H](COc23)c2ccc(Cl)cc2)ncc1\C=C(/C)C(O)=O

InChI Key InChIKey=PVBKEJLCGWHLIX-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 556452   

TargetGlucagon-like peptide 1 receptor(Human)
Gasherbrum Bio

US Patent
LigandPNGBDBM556452(US11897851, Compound 208a)
Affinity DataEC50:  0.0110nMAssay Description:To optimize functional activity directed toward Gas coupling, a HEK293/CRE-Luc cell line developed by HDB stably expressing the GLP-1 Receptor was us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/17/2024
Entry Details
US Patent