BDBM570765 US11440886, Example 101-2::US11440886, Example 98-2

SMILES Cc1cc(=O)cc(C)n1\C=C\c1ccc(OC(F)F)c(O[C@H]2CC[S@@+]([O-])C2)c1

InChI Key InChIKey=DUDOVLKRJONDFE-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 570765   

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
E-Nitiate Biopharmaceuticals (Hangzhou)

US Patent
LigandPNGBDBM570765(US11440886, Example 101-2 | US11440886, Example 98...)
Affinity DataIC50: 12.5nMAssay Description:The inhibitory effect of the compounds on human PDE4B1 enzyme activity was determined by quantifying the 5′-adenosine monophosphate (5′-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent

TargetcAMP-specific 3',5'-cyclic phosphodiesterase 4B(Human)
E-Nitiate Biopharmaceuticals (Hangzhou)

US Patent
LigandPNGBDBM570765(US11440886, Example 101-2 | US11440886, Example 98...)
Affinity DataIC50: 26nMAssay Description:The inhibitory effect of the compounds on human PDE4B1 enzyme activity was determined by quantifying the 5′-adenosine monophosphate (5′-A...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/19/2022
Entry Details
US Patent