BDBM577096 8-Cyclopropyl-10-(4-methylphenyl)pyrido[2′,3′:4,5]pyrrolo[1,2-a]pyrazin-9(8H)-one ::US11472805, Example 13
SMILES Cc1ccc(cc1)-c1c2ncccc2n2ccn(C3CC3)c(=O)c12
InChI Key InChIKey=AVBSGRYHZMSEHV-UHFFFAOYSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 577096
Affinity DataIC50: 1.86nMAssay Description:The PDE4A3, PDE4B1, PDE4C1 and PDE4D3 assays use the Scintillation Proximity Assay (SPA) technology to measure the inhibition of human recombinant PD...More data for this Ligand-Target Pair
TargetIsoform 3 of cAMP-specific 3',5'-cyclic phosphodiesterase 4D (hPDE4D3) [50-672](Human)
Pfizer
US Patent
Pfizer
US Patent