BDBM608087 (1-cyclopropyl-1H-imidazol-4-yl)[(1R,5S,6r)-6-(5,5-dimethyl-4,5-dihydro-1,2-oxazol-3-yl)-6-methyl-3-azabicyclo[3.1.0]hex-3-yl]methanone::US11691968, Example 82::US20230271952, Example 82

SMILES C[C@]1([C@H]2CN(C[C@@H]12)C(=O)c1cn(cn1)C1CC1)C1=NOC(C)(C)C1

InChI Key InChIKey=YTBUTMFDMVPZNY-MCBXIFIFSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 608087   

TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM608087((1-cyclopropyl-1H-imidazol-4-yl)[(1R,5S,6r)-6-(5,5...)
Affinity DataIC50:  30nMAssay Description:Using 384-well white Greiner784075 (Greiner), representative compounds were characterized for their inhibition of KDM5A using HTRF technology (Cisbio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM608087((1-cyclopropyl-1H-imidazol-4-yl)[(1R,5S,6r)-6-(5,5...)
Affinity DataIC50:  30nMAssay Description:Using 384-well white Greiner784075 (Greiner), representative compounds were characterized for their inhibition of KDM5A using HTRF® technology (Cisbi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent