BDBM608091 US11691968, Example 88::US20230271952, Example 88::[(1R,5S,6r)-6-(5,5-dimethyl-4,5-dihydro-1,2-oxazol-3-yl)-3-azabicyclo[3.1.0]hex-3-yl](5-isopropyl-1H-pyrazol-3-yl)methanone

SMILES CC(C)c1cc(n[nH]1)C(=O)N1C[C@H]2[C@@H](C1)[C@@H]2C1=NOC(C)(C)C1

InChI Key

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 608091   

TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM608091(US11691968, Example 88 | US20230271952, Example 88...)
Affinity DataIC50:  70nMAssay Description:Using 384-well white Greiner784075 (Greiner), representative compounds were characterized for their inhibition of KDM5A using HTRF technology (Cisbio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
Ono Pharmaceutical

US Patent
LigandPNGBDBM608091(US11691968, Example 88 | US20230271952, Example 88...)
Affinity DataIC50:  70nMAssay Description:Using 384-well white Greiner784075 (Greiner), representative compounds were characterized for their inhibition of KDM5A using HTRF® technology (Cisbi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent