BDBM611067 1-(3-Chloro-2-methylindazol-5-yl)-2- (4-cyano-3-fluorophenyl)-N-[(3R)-1- methylpiperidin-3-yl]imidazole-4- carboxamide::US10626103, Example 59

SMILES CN1CCC[C@H](C1)NC(=O)c1cn(c(n1)-c1ccc(C#N)c(F)c1)-c1ccc2nn(C)c(Cl)c2c1

InChI Key InChIKey=LIMDPDHBURVMDW-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 611067   

TargetLysine-specific histone demethylase 1A(Human)
Celgene Quanticel Research

US Patent
LigandPNGBDBM611067(US10626103, Example 59 | 1-(3-Chloro-2-methylindaz...)
Affinity DataIC50: 100nMAssay Description:The enzymatic assay of LSD1 activity is based on Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The inhibitory properties ...More data for this Ligand-Target Pair
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Date in BDB:
9/8/2023
Entry Details
US Patent