BDBM614900 US20230271937, Example A7-57

SMILES CCN(Cc1ccc(cc1)C(F)(F)F)c1ncnc(NC[C@@H]2CCN(C[C@H]2O)C(C)(C)C(N)=O)c1F

InChI Key InChIKey=PQRWVUIEJYNURD-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 614900   

TargetPeroxisome proliferator-activated receptor gamma(Human)
Nuevolution

US Patent
LigandPNGBDBM614900(US20230271937, Example A7-57)
Affinity DataEC50:  7.90nMAssay Description:The HEK293 cell line is co-transfected transiently with two plasmids, one with the RORγ ligand-binding domain fused to galactose-responsive tran...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
US Patent