BDBM615101 US20230271949, Example 2

SMILES O[C@@H]1C[C@H](N(C1)C(=O)CNC(=O)c1ccc2n(CC3CCO3)c(CN3CCC(CC3)c3cccc(OCc4ccc(Cl)cc4F)n3)nc2c1)C(O)=O

InChI Key InChIKey=QOCYISJFQNNAPV-UHFFFAOYSA-N

Data  1 KI  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 615101   

TargetGlucagon-like peptide 1 receptor(Human)
Ascletis Bioscience

US Patent
LigandPNGBDBM615101(US20230271949, Example 2)
Affinity DataEC50:  0.320nMAssay Description:cAMP Detection Kit, Cisbio (Cat #62AM4PEJ).More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
US Patent

TargetGlucagon-like peptide 1 receptor(Human)
Ascletis Bioscience

US Patent
LigandPNGBDBM615101(US20230271949, Example 2)
Affinity DataKi:  165nMAssay Description:Tag-Lite Binding Assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
US Patent

TargetGlucagon-like peptide 1 receptor(Human)
Ascletis Bioscience

US Patent
LigandPNGBDBM615101(US20230271949, Example 2)
Affinity DataIC50: 345nMAssay Description:Tag-Lite Binding Assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
US Patent