BDBM615163 US20230271949, Example 5

SMILES Cc1n[nH]c2ccc(NC(=O)c3ccc4n(C[C@@H]5CCO5)c(CN5CCC(=CC5)c5cccc6O[C@@](C)(Oc56)c5ccc(Cl)cc5F)nc4c3)cc12

InChI Key InChIKey=MOLZPTPRJQOUDS-UHFFFAOYSA-N

Data  1 KI  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 615163   

TargetGlucagon-like peptide 1 receptor(Human)
Ascletis Bioscience

US Patent
LigandPNGBDBM615163(US20230271949, Example 5)
Affinity DataEC50:  0.120nMAssay Description:cAMP Detection Kit, Cisbio (Cat #62AM4PEJ).More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
US Patent

TargetGlucagon-like peptide 1 receptor(Human)
Ascletis Bioscience

US Patent
LigandPNGBDBM615163(US20230271949, Example 5)
Affinity DataKi:  911nMAssay Description:Tag-Lite Binding Assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
US Patent

TargetGlucagon-like peptide 1 receptor(Human)
Ascletis Bioscience

US Patent
LigandPNGBDBM615163(US20230271949, Example 5)
Affinity DataIC50: 1.71E+3nMAssay Description:Tag-Lite Binding Assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
US Patent