BDBM615412 US20230271949, Example 203

SMILES Fc1cc(Cl)ccc1COc1cccc(n1)C1=CCN(Cc2nc3cc(NC(=O)c4ccc5NC(=O)C6(CC6)c5c4)ccc3n2C[C@@H]2CCO2)CC1

InChI Key InChIKey=UXQHCUIXAUEOSD-UHFFFAOYSA-N

Data  1 KI  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 615412   

TargetGlucagon-like peptide 1 receptor(Human)
Ascletis Bioscience

US Patent
LigandPNGBDBM615412(US20230271949, Example 203)
Affinity DataEC50:  0.240nMAssay Description:cAMP Detection Kit, Cisbio (Cat #62AM4PEJ).More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
US Patent

TargetGlucagon-like peptide 1 receptor(Human)
Ascletis Bioscience

US Patent
LigandPNGBDBM615412(US20230271949, Example 203)
Affinity DataKi:  90.3nMAssay Description:Tag-Lite Binding Assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
US Patent

TargetGlucagon-like peptide 1 receptor(Human)
Ascletis Bioscience

US Patent
LigandPNGBDBM615412(US20230271949, Example 203)
Affinity DataIC50: 158nMAssay Description:Tag-Lite Binding Assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/15/2023
Entry Details
US Patent