BDBM618970 US20230295110, Compound 4.

SMILES Cc1c(O)c(ncc1-c1cnn(c1)-c1ccccc1)C(=O)NCC(O)=O

InChI Key InChIKey=ADZOKWWFAGEXFM-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 618970   

TargetProlyl hydroxylase EGLN2(Human)
Akebia Therapeutics

US Patent
LigandPNGBDBM618970(US20230295110, Compound 4.)
Affinity DataIC50: 100nMAssay Description:Time-resolved fluorescence resonance energy transfer (TR-FRET) assay was utilized to determine the enzymatic half maximal inhibitory concentration (I...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent

TargetEgl nine homolog 1(Human)
Akebia Therapeutics

US Patent
LigandPNGBDBM618970(US20230295110, Compound 4.)
Affinity DataIC50: 100nMAssay Description:Time-resolved fluorescence resonance energy transfer (TR-FRET) assay was utilized to determine the enzymatic half maximal inhibitory concentration (I...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2023
Entry Details
US Patent