BDBM629024 N-(4-(3-(5-Fluoropyridin-2-yl)-1-methyl-1H-pyrazol-4-yl)pyridin-2-yl)::US20230339900, Example 1

SMILES CCC(=O)Nc1cc(ccn1)-c1cn(C)nc1-c1ccc(F)cn1

InChI Key InChIKey=GCGRJPHGTHHQEX-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 629024   

TargetCasein kinase I isoform delta(Human)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM629024(US20230339900, Example 1 | N-(4-(3-(5-Fluoropyridi...)
Affinity DataIC50: 107nMAssay Description:In this assay, CSNK1D phosphorylates a substrate peptide PLSRTL-pS-VASLPGL in the presence of ATP. This substrate peptide has been modeled after the ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2023
Entry Details
US Patent