BDBM629103 4-[3-(5-Fluoro-2-pyridyl)-1-methyl-pyrazol-4-yl]-6-methyl-1H-pyrrolo[2,3-b]::US20230339900, Example 80

SMILES Cc1cc(-c2cn(C)nc2-c2ccc(F)cn2)c2cc[nH]c2n1

InChI Key InChIKey=HBQHSHVNQVPPJF-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 629103   

TargetCasein kinase I isoform delta(Human)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM629103(US20230339900, Example 80 | 4-[3-(5-Fluoro-2-pyrid...)
Affinity DataIC50: 41nMAssay Description:In this assay, CSNK1D phosphorylates a substrate peptide PLSRTL-pS-VASLPGL in the presence of ATP. This substrate peptide has been modeled after the ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2023
Entry Details
US Patent