BDBM639405 (cyclobutylmethyl)({2- [(4-{1- fluoroimidazo[1,5- a]pyridin-8-yl}-1H- 1,2,3-triazol-1- yl)methyl]imidazo [1,2-a]pyridin-6- yl}methyl)amine::US20230391770, Example 25

SMILES Fc1ncn2cccc(-c3cn(Cc4cn5cc(CNCC6CCC6)ccc5n4)nn3)c12

InChI Key InChIKey=VGUJVECZZOSQLT-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 639405   

LigandPNGBDBM639405((cyclobutylmethyl)({2- [(4-{1- fluoroimidazo[1,5- ...)
Affinity DataIC50: 15.8nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2024
Entry Details
US Patent