BDBM639410 2-({2-[(4-{6- methoxyimidazo[1,5- a]pyridin-8-yl}-1H- 1,2,3-triazol-1- yl)methyl]imidazo [1,2-a]pyridin-6- yl}methyl)-2- azaspiro[3.3] heptane::US20230391770, Example 30

SMILES COc1cc(-c2cn(Cc3cn4cc(CN5CC6(CCC6)C5)ccc4n3)nn2)c2cncn2c1

InChI Key InChIKey=FEFIBVQAEIUCCS-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 639410   

LigandPNGBDBM639410(2-({2-[(4-{6- methoxyimidazo[1,5- a]pyridin-8-yl}-...)
Affinity DataIC50: 6.10nMAssay Description:The enzymatic assay was established to determine IC50 values for inhibition of RNA methyltransferase activity. The enzyme used was full-length his-ta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2024
Entry Details
US Patent