BDBM645391 US20240016810, Compound TABLE 16.4::US20240208964, Biochemistry 4

SMILES C1CN(CC(N1)c1ccccc1)c1cc(N2CCOCC2)n2nc(cc2n1)-c1ccncc1

InChI Key InChIKey=VLPBRHSABODXQH-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 645391   

LigandPNGBDBM645391(US20240016810, Compound TABLE 16.4 | US20240208964...)
Affinity DataIC50: 2.66E+3nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM645391(US20240016810, Compound TABLE 16.4 | US20240208964...)
Affinity DataIC50: 2.66E+3nMAssay Description:The biochemical PIKfyve inhibition assays were run by Carna Biosciences according to proprietary methodology based on the Promega ADP-Glo™ Kinase ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM645391(US20240016810, Compound TABLE 16.4 | US20240208964...)
Affinity DataIC50: 2.66E+3nMAssay Description:The biochemical PIKFyve inhibition assays were run by Carna Biosciences according to proprietary methodology based on the Promega ADP-Glo Kinase assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2024
Entry Details
US Patent

LigandPNGBDBM645391(US20240016810, Compound TABLE 16.4 | US20240208964...)
Affinity DataIC50: 2.66E+3nMAssay Description:The biochemical PIKFyve inhibition assays were run by Carna Biosciences according to proprietary methodology based on the Promega ADP-Glo Kinase assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

LigandPNGBDBM645391(US20240016810, Compound TABLE 16.4 | US20240208964...)
Affinity DataIC50: 1.50E+4nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent