BDBM645395 US20240016810, Compound TABLE 16.8::US20240150358, Example 00174::US20240208964, Biochemistry 8

SMILES O=c1ccc(nn1-c1cc(N2CCOCC2)n2nc(cc2n1)-c1ccncc1)-c1ccccc1

InChI Key InChIKey=PITJQADZDFCFOH-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 645395   

LigandPNGBDBM645395(US20240016810, Compound TABLE 16.8 | US20240208964...)
Affinity DataIC50: 295nMAssay Description:The biochemical PIKfyve inhibition assays were run by Carna Biosciences according to proprietary methodology based on the Promega ADP-Glo™ Kinase ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM645395(US20240016810, Compound TABLE 16.8 | US20240208964...)
Affinity DataIC50: 295nMAssay Description:The biochemical PIKFyve inhibition assays were run by Carna Biosciences according to proprietary methodology based on the Promega ADP-Glo Kinase assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/13/2024
Entry Details
US Patent

LigandPNGBDBM645395(US20240016810, Compound TABLE 16.8 | US20240208964...)
Affinity DataIC50: 295nMAssay Description:The biochemical PIKFyve inhibition assays were run by Carna Biosciences according to proprietary methodology based on the Promega ADP-Glo Kinase assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2024
Entry Details
US Patent

LigandPNGBDBM645395(US20240016810, Compound TABLE 16.8 | US20240208964...)
Affinity DataIC50: 295nMAssay Description:The biochemical PIKFyve inhibition assays were run by Carna Biosciences according to proprietary methodology based on the Promega ADP-Glo Kinase assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
US Patent

LigandPNGBDBM645395(US20240016810, Compound TABLE 16.8 | US20240208964...)
Affinity DataIC50: 295nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM645395(US20240016810, Compound TABLE 16.8 | US20240208964...)
Affinity DataIC50: 1.50E+4nMAssay Description:PIKfyve Biochemical Assay. The biochemical PIKFyve inhibition assays were run by Cama Biosciences according to proprietary methodology based on the P...More data for this Ligand-Target Pair
In Depth
Date in BDB:
TBA
Entry Details
US Patent