BDBM652296 US20240058459, Compound D-didesethyl Sunitinib conjugate (D-4517)

SMILES COC(=O)CCC\C(N)=C\NCCOCCOCCOCCC(=O)NCCNC(=O)c1c(C)nc(\C=C2/C(=O)Nc3ccc(F)cc23)c1C

InChI Key

Data  1 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 652296   

TargetVascular endothelial growth factor receptor 2(Human)
Ashvattha Therapeutics

US Patent
LigandPNGBDBM652296(US20240058459, Compound D-didesethyl Sunitinib con...)
Affinity DataKd:  27nMAssay Description:Kinase-tagged T7 phage strains were prepared in an E. coli host derived from the BL21 strain. E. coli were grown to log-phase and infected with T7 ph...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent