BDBM654842 1-(propan-2-yl)-5-{3-[3- (trifluoromethyl)pyridin-4-yl]-1,2,4- oxadiazol-5-yl}-1H-1,2,3- benzotriazole::US11912693, Compound 455
SMILES CC(C)n1nnc2cc(ccc12)-c1nc(no1)-c1ccncc1C(F)(F)F
InChI Key InChIKey=VMIDOGQVIOBXMI-UHFFFAOYSA-N
Data 4 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 654842
Affinity DataEC50: <316nMAssay Description:Agonist-promoted G-protein responses were determined by measuring changes in intracellular cAMP using the HTRF cAMP HiRange kit (CisBio, Cat #: 62AM6...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:S1P2 Agonist-promoted G-protein responses were determined by measuring changes in intracellular inositol monophosphate using the IP-one TB kit (CisBi...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist-promoted G-protein responses were determined by measuring changes in intracellular cAMP using the HTRF cAMP HiRange kit (CisBio, Cat #: 62AM6...More data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+4nMAssay Description:Agonist-promoted β-arrestin2 recruitment to the sphingosine-1-phosphate 1 receptor was determined using the β-arrestin PathHunter ) Detecti...More data for this Ligand-Target Pair