BDBM667073 7-(5-chloro-2-fluorophenyl)-1-{1H- pyrrolo[2,3- b]pyridin-4-yl}-1H,2H,3H- pyrido[3,4-b][1,4]oxazine::US20240116947, Example 16

SMILES Fc1ccc(Cl)cc1-c1cc2N(CCOc2cn1)c1ccnc2[nH]ccc12

InChI Key InChIKey=VZBWDHLVWPQRRX-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 667073   

TargetTGF-beta receptor type-1(Human)
CHIESI FARMACEUTICI S.P.A.

US Patent
LigandPNGBDBM667073(7-(5-chloro-2-fluorophenyl)-1-{1H- pyrrolo[2,3- b]...)
Affinity DataIC50: <1nMAssay Description:The enzymatic activity of compounds of the present invention was monitored measuring the formation of ADP using the ADP-GLO Kinases assay. Following ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent