BDBM681943 US20240199649, Compound 986

SMILES C[C@]1(O)CC[C@@H](CC1)Nc1nc(N)c2c(ccn2n1)-c1ccc2ncn(CC(F)F)c2n1

InChI Key InChIKey=WCKXOSRZFBVUIX-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 681943   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Biosplice Therapeutics

US Patent
LigandPNGBDBM681943(US20240199649, Compound 986)
Affinity DataIC50: 0.700nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Division ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
US Patent