BDBM683193 4-(5-((3- aminopropyl) (methyl) amino)-8-(3- hydroxy-4- methylphenyl) imidazolo[1,2-c] pyrimidin-7-yl)-2- fluorobenzonitrile::US20240216357, Example 146

SMILES CN(CCCN)c1nc(-c2ccc(C#N)c(F)c2)c(-c2ccc(C)c(O)c2)c2nccn12

InChI Key InChIKey=PFSVFLIPIZNXPF-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 683193   

TargetLysine-specific histone demethylase 1A(Human)
Sichuan Huiyu Pharmaceutical Co.

US Patent
LigandPNGBDBM683193(US20240216357, Example 146 | 4-(5-((3- aminopropyl...)
Affinity DataIC50: 0.5nMAssay Description:The effects of compounds on LSD1 enzyme activity are detected by an HTRF technology to evaluate their inhibition levels on LSD1 enzyme activity. Firs...More data for this Ligand-Target Pair
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Date in BDB:
10/11/2024
Entry Details
US Patent