BDBM683202 4-(5-(3-amino-8- azabicyclo[3.2.1] octane-8-yl)-8- (3-hydroxy-4- methylphenyl) imidazolo[1,2-c] pyrimidin-7-yl)- 2-fluorobenzo nitrile hydrochloride::US20240216357, Example 156

SMILES Cc1ccc(cc1O)-c1c(nc(N2C3CCC2CC(N)C3)n2ccnc12)-c1ccc(C#N)c(F)c1

InChI Key InChIKey=XABWFOAWLSTPRM-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 683202   

TargetLysine-specific histone demethylase 1A(Human)
Sichuan Huiyu Pharmaceutical Co.

US Patent
LigandPNGBDBM683202(US20240216357, Example 156 | 4-(5-(3-amino-8- azab...)
Affinity DataIC50: 0.200nMAssay Description:The effects of compounds on LSD1 enzyme activity are detected by an HTRF technology to evaluate their inhibition levels on LSD1 enzyme activity. Firs...More data for this Ligand-Target Pair
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Date in BDB:
10/11/2024
Entry Details
US Patent