BDBM690384 2,5-dichloro-N-[2,6- difluoro-4-(2 phenylethynyl)phenyl] benzenesulfonamide::US12065399, Example 4

SMILES Fc1cc(cc(F)c1NS(=O)(=O)c1cc(Cl)ccc1Cl)C#Cc1ccccc1

InChI Key InChIKey=FTDRNDFGKHVRKT-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 690384   

TargetMetabotropic glutamate receptor 4(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM690384(US12065399, Example 4 | 2,5-dichloro-N-[2,6- diflu...)
Affinity DataEC50:  3.43E+3nMAssay Description:A monoclonal HEK-293 cell line stably transfected with a cDNA encoding for the human mGlu4 receptor was generated. Cells were cultured according to s...More data for this Ligand-Target Pair
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Date in BDB:
11/26/2024
Entry Details
US Patent