BDBM691220 (R)-N-(5-(5-ethyl-1,2,4-oxadiazol-3- yl)-7-hydroxy-2,3-dihydro-1H-inden- 1-yl)-1-methyl-1H-pyrazole-4- carboxamide::US12065436, Compound 609

SMILES CCc1nc(no1)-c1cc2CC[C@@H](NC(=O)c3cnn(C)c3)c2c(O)c1

InChI Key InChIKey=QSNUZRFMGOSWJQ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 691220   

TargetMyosin-1(Bovine)
Cytokinetics

US Patent
LigandPNGBDBM691220(US12065436, Compound 609 | (R)-N-(5-(5-ethyl-1,2,4...)
Affinity DataIC50: 900nMAssay Description:To evaluate the effect of compounds on the ATPase activity of full-length cardiac myosin in the context of the native sarcomere, skinned myofibril as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2024
Entry Details
US Patent