BDBM691258 (R)-2-chloro-N-(5-(5-ethyl-1,2,4- oxadiazol-3-yl)-2,3-dihydro-1H- inden-1-yl)isonicotinamide::US12065436, Compound 647

SMILES CCc1nc(no1)-c1ccc2[C@@H](CCc2c1)NC(=O)c1ccnc(Cl)c1

InChI Key InChIKey=IFRGDCLAVFIWSR-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 691258   

TargetMyosin-1(Bovine)
Cytokinetics

US Patent
LigandPNGBDBM691258(US12065436, Compound 647 | (R)-2-chloro-N-(5-(5-et...)
Affinity DataIC50: 900nMAssay Description:To evaluate the effect of compounds on the ATPase activity of full-length cardiac myosin in the context of the native sarcomere, skinned myofibril as...More data for this Ligand-Target Pair
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Date in BDB:
11/26/2024
Entry Details
US Patent