BDBM695809 2-((8-Chloro-1-(2,6-dichloro-4-(2-hydroxyethoxy)phenyl)-2-methyl-4-oxo-1,4-dihydro-1,6-naphthyridin-5-yl)oxy)-N-(2-hydroxyethyl)acetamide ::US12084442, Example 2

SMILES Cc1cc(=O)c2c(OCC(=O)NCCO)ncc(Cl)c2n1-c1c(Cl)cc(OCCO)cc1Cl

InChI Key InChIKey=KTECXOYSCVMAJD-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 695809   

LigandPNGBDBM695809(US12084442, Example 2 | 2-((8-Chloro-1-(2,6-dichlo...)
Affinity DataIC50: 220nMAssay Description:The GIRK1/4 activity of a compound according to the present invention was assessed by the following in vitro method.Buffers:a. External buffer: 10 mM...More data for this Ligand-Target Pair
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Date in BDB:
1/6/2025
Entry Details
US Patent