BDBM695816 N-(2-((8-chloro-1-(2,6-dichloro-4-(2-hydroxyethoxy)phenyl)-2-methyl-4-oxo-1,4-dihydro-1,6-naphthyridin-5-yl)oxy)ethyl)acetamide ::US12084442, Example 9

SMILES CC(=O)NCCOc1ncc(Cl)c2n(c(C)cc(=O)c12)-c1c(Cl)cc(OCCO)cc1Cl

InChI Key InChIKey=VRJVSLVXQLHPQC-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 695816   

LigandPNGBDBM695816(US12084442, Example 9 | N-(2-((8-chloro-1-(2,6-dic...)
Affinity DataIC50: 80nMAssay Description:The GIRK1/4 activity of a compound according to the present invention was assessed by the following in vitro method.Buffers:a. External buffer: 10 mM...More data for this Ligand-Target Pair
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Date in BDB:
1/6/2025
Entry Details
US Patent