BDBM695824 2-(4-(5-(2-Amino-2-oxoethoxy)-8-chloro-2-methyl-4-oxo-1,6-naphthyridin-1(4H)-yl)-3,5-dichlorophenoxy)-N-methylacetamide ::US12084442, Example 17

SMILES CNC(=O)COc1cc(Cl)c(c(Cl)c1)-n1c(C)cc(=O)c2c(OCC(N)=O)ncc(Cl)c12

InChI Key InChIKey=IUNMBOLIOPFUTE-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 695824   

LigandPNGBDBM695824(US12084442, Example 17 | 2-(4-(5-(2-Amino-2-oxoeth...)
Affinity DataIC50: 250nMAssay Description:The GIRK1/4 activity of a compound according to the present invention was assessed by the following in vitro method.Buffers:a. External buffer: 10 mM...More data for this Ligand-Target Pair
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Date in BDB:
1/6/2025
Entry Details
US Patent