BDBM697082 US20240309004, Compound VKT-034

SMILES N[C@@H]1CCC(C1)Nc1cc2c3ccc(F)cc3nn2cn1

InChI Key InChIKey=QJTSTYYTCWCYDQ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 697082   

TargetCyclin-T1/Cyclin-dependent kinase 9(Human)
Virokyne Therapeutics

US Patent
LigandPNGBDBM697082(US20240309004, Compound VKT-034)
Affinity DataIC50: 80.7nMAssay Description:Compounds VKT-007, VKT-034, VKT-036, and VKT-511 were tested in 10-dose IC50 duplicate mode with a 3-fold serial dilution starting at 10 μM. Con...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
1/16/2025
Entry Details
US Patent

TargetCyclin-H/Cyclin-dependent kinase 7(Human)
Virokyne Therapeutics

US Patent
LigandPNGBDBM697082(US20240309004, Compound VKT-034)
Affinity DataIC50: 2.54E+3nMAssay Description:Compounds VKT-007, VKT-034, VKT-036, and VKT-511 were tested in 10-dose IC50 duplicate mode with a 3-fold serial dilution starting at 10 μM. Con...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
1/16/2025
Entry Details
US Patent