BDBM701173 4-[2-(N-cyclohexylanilino)-2-oxo-ethyl]-1- [cyclopropyl-(4- fluorophenyl)carbamoyl]piperidine-4- carboxylic acid::US12122750, Example 16

SMILES O=C(CC1(C(=O)O)CCN(C(=O)N(c2ccc(F)cc2)C2CC2)CC1)N(c1ccccc1)C1CCCCC1

InChI Key InChIKey=RVZKYVOXSPRMMZ-UHFFFAOYSA-N

Data  1 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 701173   

TargetType-2 angiotensin II receptor(Human)
Eli Lilly

US Patent
LigandPNGBDBM701173(4-[2-(N-cyclohexylanilino)-2-oxo-ethyl]-1- [cyclop...)
Affinity DataKi:  1.76nMAssay Description:Receptor binding affinities (Ki) were determined from a competitive radioligand binding assay with human recombinant ([125I]-Tyr4)-Angiotensin-II (22...More data for this Ligand-Target Pair
Ligand InfoSimilars
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Date in BDB:
2/24/2025
Entry Details
US Patent