BDBM708491 3-(2-methyl-5-(8-(4- methylpiperazin-1- yl)oct-1-yn-1-yl)- 4-oxoquinazolin-3(4H)- yl)piperidine-2,6-dione::US20240425475, Compound GT-02645

SMILES Cc1nc2cccc(C#CCCCCCCN3CCN(C)CC3)c2c(=O)n1C1CCC(=O)NC1=O

InChI Key InChIKey=RKROHFOPAOBOOC-UHFFFAOYSA-N

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 708491   

TargetProtein cereblon(Human)
Gluetacs Therapeutics (Shanghai) Co.

US Patent
LigandPNGBDBM708491(3-(2-methyl-5-(8-(4- methylpiperazin-1- yl)oct-1-y...)
Affinity DataIC50: 2.80E+3nMAssay Description:1. According to the instructions of the CEREBLON BINDING kits, the compounds to be tested of the present invention and lenalidomide were serially dil...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/7/2025
Entry Details
US Patent