BDBM709097 tert-butyl-N-{2-[({2-methoxy-5-[3-(methylcarbamoyl)-1H-indazol-6-yl]pyridin-3-yl}-formamido)methyl]phenyl}-carbamate::US12172975, Example 73

SMILES CNC(=O)c1n[nH]c2cc(-c3cnc(OC)c(C(=O)NCc4ccccc4NC(=O)OC(C)(C)C)c3)ccc12

InChI Key InChIKey=DAAKIMHMUVUXIU-UHFFFAOYSA-N

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 709097   

TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM709097(tert-butyl-N-{2-[({2-methoxy-5-[3-(methylcarbamoyl...)
Affinity DataIC50: 4.70nMAssay Description:A solution was prepared containing 0.2 nM Anti GST-Tb (Cisbio, 61GSTTLB), 90.6 nM probe and 1 nM His-GST-TVMV-hRIPK1 (1-324) in FRET Buffer (20 mM HE...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/5/2025
Entry Details
US Patent