BDBM712424 4-((2-(4-((4-(((2-(2,6-Dioxopiperidin-3-yl)-1,3-dioxoisoindolin-4-yl)amino)methyl)-1H-1,2,3-triazol-1-yl)methyl)phenyl)-7-phenylimidazo[1,2-a]pyridin-3-yl)amino)benzoic acid::US20250011330, Compound XZ747

SMILES O=C1CCC(N2C(=O)c3cccc(NCc4cn(Cc5ccc(-c6nc7cc(-c8ccccc8)ccn7c6Nc6ccc(C(=O)O)cc6)cc5)nn4)c3C2=O)C(=O)N1

InChI Key InChIKey=FZNOVWFLSRQHEM-UHFFFAOYSA-N

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 712424   

TargetTyrosyl-DNA phosphodiesterase 1(Human)
Department Of Health and Human Services

US Patent
LigandPNGBDBM712424(4-((2-(4-((4-(((2-(2,6-Dioxopiperidin-3-yl)-1,3-di...)
Affinity DataIC50: 7.41E+3nMAssay Description:The oximes were evaluated by gel-based TDP1 fluorescence assay in a concentration of 100 μM in DMSO. The fluorescence of DMSO blank vial was set as 0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/22/2025
Entry Details
US Patent

TargetTyrosyl-DNA phosphodiesterase 2(Human)
Department Of Health and Human Services

US Patent
LigandPNGBDBM712424(4-((2-(4-((4-(((2-(2,6-Dioxopiperidin-3-yl)-1,3-di...)
Affinity DataIC50: 1.12E+4nMAssay Description:The oximes were evaluated by gel-based TDP1 fluorescence assay in a concentration of 100 μM in DMSO. The fluorescence of DMSO blank vial was set as 0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/22/2025
Entry Details
US Patent