BDBM713962 US12202839, Compound 9k

SMILES N=C1C(=O)NC(=O)c2cc(-c3ccccc3Cl)sc21

InChI Key InChIKey=DXWKXJCHISYLMA-UHFFFAOYSA-N

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 713962   

TargetProtein tyrosine phosphatase type IVA 3(Human)
University of Virginia Patent Foundation

US Patent
LigandPNGBDBM713962(US12202839, Compound 9k)
Affinity DataIC50: 36.1nMAssay Description:Enzyme activity assays were performed in triplicate in 384-well Greiner Bio-One black small volume microtiter plates, as previously described using r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
US Patent

TargetProtein tyrosine phosphatase type IVA 3(Human)
University of Virginia Patent Foundation

US Patent
LigandPNGBDBM713962(US12202839, Compound 9k)
Affinity DataIC50: 36.1nMAssay Description:Table 4: In Vitro Biochemical Analysis of PTP4A Inhibition. Enzyme activity assays were performed in triplicate in 384-well Greiner Bio-One black sma...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
US Patent

TargetProtein tyrosine phosphatase type IVA 3(Human)
University of Virginia Patent Foundation

US Patent
LigandPNGBDBM713962(US12202839, Compound 9k)
Affinity DataIC50: 36.1nMAssay Description:Enzyme activity assays were performed in triplicate in 384-well Greiner Bio-One black small volume microtiter plates, as previously described using r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
US Patent

TargetProtein tyrosine phosphatase type IVA 3(Human)
University of Virginia Patent Foundation

US Patent
LigandPNGBDBM713962(US12202839, Compound 9k)
Affinity DataIC50: 36.1nMAssay Description:Table 2: Recombinant human PTP4A3 phosphatase was used and the enzymatic assay was performed as previously described,20 except that it was fully auto...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
US Patent

TargetProtein tyrosine phosphatase type IVA 1(Human)
University of Virginia Patent Foundation

US Patent
LigandPNGBDBM713962(US12202839, Compound 9k)
Affinity DataIC50: 49nMAssay Description:Enzyme activity assays were performed in triplicate in 384-well Greiner Bio-One black small volume microtiter plates, as previously described using r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
US Patent

TargetProtein tyrosine phosphatase type IVA 1(Human)
University of Virginia Patent Foundation

US Patent
LigandPNGBDBM713962(US12202839, Compound 9k)
Affinity DataIC50: 49nMAssay Description:Table 4: In Vitro Biochemical Analysis of PTP4A Inhibition. Enzyme activity assays were performed in triplicate in 384-well Greiner Bio-One black sma...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
US Patent

TargetProtein tyrosine phosphatase type IVA 2(Human)
University of Virginia Patent Foundation

US Patent
LigandPNGBDBM713962(US12202839, Compound 9k)
Affinity DataIC50: 113nMAssay Description:Enzyme activity assays were performed in triplicate in 384-well Greiner Bio-One black small volume microtiter plates, as previously described using r...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
US Patent

TargetProtein tyrosine phosphatase type IVA 2(Human)
University of Virginia Patent Foundation

US Patent
LigandPNGBDBM713962(US12202839, Compound 9k)
Affinity DataIC50: 113nMAssay Description:Table 4: In Vitro Biochemical Analysis of PTP4A Inhibition. Enzyme activity assays were performed in triplicate in 384-well Greiner Bio-One black sma...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
US Patent