BDBM717689 US12215173, Compound DAMGO

SMILES C[C@@H](NC(=O)CCc1ccc(O)cc1)C(=O)NCC(=O)N(C)[C@@H](Cc1ccccc1)C(=O)NCCO

InChI Key InChIKey=SFHAPPCUMVWDSX-UHFFFAOYSA-N

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 717689   

TargetMu-type opioid receptor(Human)
Humanwell Pharmaceutical US

US Patent
LigandPNGBDBM717689(US12215173, Compound DAMGO)
Affinity DataIC50: 0.426nMAssay Description:The assay buffers used for opioid receptor binding studies were 50 mM Tris HCl (pH 7.4) for KOR, 50 mM Tris HCl (pH 7.4) with 5 mM MgCl2 for MOR, and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/10/2025
Entry Details
US Patent