BDBM720166 6-({5-methyl-3-[6-(trifluoromethyl)pyridin-3-yl]-1,2-oxazol-4-yl}methoxy)-2-(oxan-4-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine::US20250051323, Example 7

SMILES Cc1onc(-c2ccc(C(F)(F)F)nc2)c1COc1cc2c(cn1)CN(C1CCOCC1)CC2

InChI Key InChIKey=AEJSRKGGRHHMDY-UHFFFAOYSA-N

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 720166   

TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Human)
Richter Gedeon

US Patent
LigandPNGBDBM720166(6-({5-methyl-3-[6-(trifluoromethyl)pyridin-3-yl]-1...)
Affinity DataKi:  29.3nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampule of membrane homogenate was thawed and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
US Patent