BDBM722832 US20250059214, Compound 6

SMILES Cc1nc(C)c(C(=O)N[C@H](CC(=O)N2CCOCC2)C(=O)N[C@@H](CC(C)C)B(O)O)o1

InChI Key InChIKey=QRDCWUXUSGLJHF-UHFFFAOYSA-N

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 722832   

TargetLon protease homolog, mitochondrial(Human)
Pretzel Therapeutics

US Patent
LigandPNGBDBM722832(US20250059214, Compound 6)
Affinity DataIC50: 275nMAssay Description:In this Example, LONP1 (NM_004793.4) activity was measured by a FRET-based assay for protease activity using a fluorogenic peptide DabcylYRGIT(2Abu)S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/19/2025
Entry Details
US Patent