BDBM722872 US20250059214, Compound 48

SMILES O=C(N[C@@H](CCCc1ccccc1)B(O)O)[C@@H](CC(=O)N1CCOCC1)NC(=O)[C@H]1CCCCO1

InChI Key InChIKey=MFEFTMRFRSEKHT-UHFFFAOYSA-N

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 722872   

TargetLon protease homolog, mitochondrial(Human)
Pretzel Therapeutics

US Patent
LigandPNGBDBM722872(US20250059214, Compound 48)
Affinity DataIC50: 275nMAssay Description:In this Example, LONP1 (NM_004793.4) activity was measured by a FRET-based assay for protease activity using a fluorogenic peptide DabcylYRGIT(2Abu)S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/19/2025
Entry Details
US Patent