BDBM724704 3-methyl-N-((1r,3r)- 3-morpholinocyclo- butyl)-1-neopentyl- 1H-thieno[2,3-c]pyr- azole-5-carboxamide::US20250066383, Compound II-25

SMILES Cc1nn(CC(C)(C)C)c2sc(C(=O)N[C@H]3C[C@H](N4CCOCC4)C3)cc12

InChI Key InChIKey=OBYAKFOFMIAQAB-UHFFFAOYSA-N

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 724704   

LigandPNGBDBM724704(3-methyl-N-((1r,3r)- 3-morpholinocyclo- butyl)-1-n...)
Affinity DataIC50: 20nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandPNGBDBM724704(3-methyl-N-((1r,3r)- 3-morpholinocyclo- butyl)-1-n...)
Affinity DataIC50: 65nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent