BDBM724713 N-((1r,3r)-3-(4-cyclo- propylpiperazin-1- yl)cyclobutyl)-3- methyl-1-neopentyl- 1H-thieno[2,3-c] pyrazole-5-carbox- amide::US20250066383, Compound II-34

SMILES Cc1nn(CC(C)(C)C)c2sc(C(=O)N[C@H]3C[C@H](N4CCN(C5CC5)CC4)C3)cc12

InChI Key InChIKey=XZJXDMHVKZMWSI-UHFFFAOYSA-N

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 724713   

LigandPNGBDBM724713(N-((1r,3r)-3-(4-cyclo- propylpiperazin-1- yl)cyclo...)
Affinity DataIC50: 20nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent

LigandPNGBDBM724713(N-((1r,3r)-3-(4-cyclo- propylpiperazin-1- yl)cyclo...)
Affinity DataIC50: 65nMAssay Description:Compounds were tested for their activity by measuring the inhibition of PDE7A or PDE7B hydrolysis of [3H]cAMP to [3H]AMP. Generally, eight dilutions ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/30/2025
Entry Details
US Patent