BDBM725742 US20250074910, Example 42-1

SMILES [2H]C([2H])([2H])C1C[C@]2(CC[C@@H](CN3CCC4(CC3)CN(c3ncnnc3Oc3ccc(F)cc3C(=O)N(CC)C(C)C)C4)CC2)CC1=O

InChI Key InChIKey=GUYWJFAJILNOPJ-GKOSEXJESA-N

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 725742   

TargetHistone-lysine N-methyltransferase 2A(Human)
Hitgen

US Patent
LigandPNGBDBM725742(US20250074910, Example 42-1)
Affinity DataIC50: 15.3nMAssay Description:The inhibition of Menin/MLL-4-43 peptide interaction by small molecule inhibitors was quantitatively detected by fluorescence polarization competitio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/9/2025
Entry Details
US Patent